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【结 构 式】 
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【分子编号】69618 【品名】(6R,7R)-7-amino-3-(hydroxymethyl)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid 【CA登记号】 |
【 分 子 式 】C8H10N2O4S 【 分 子 量 】230.24448 【元素组成】C 41.73% H 4.38% N 12.17% O 27.8% S 13.93% |
与该中间体有关的原料药合成路线共 1 条
合成路线1
该中间体在本合成路线中的序号：(II)
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| 【3】 程清蓉，刘志雄，李翔，等.去甲氨噻肟酸乙酯的合成研究.化学世界，2007,48:480 |
| 【4】 郑庚修，李贺，赵叶青.制备去甲氨噻肟酸乙酯的方法：CN,Patent 101,007,793,2007. |
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| 中间体序号 | 中间体编号 | 品名 | CAS号 | 分子式 | 供应商 | 用于合成 |
|---|---|---|---|---|---|---|
| (I) | 22747 | (6R,7R)-3-[(acetoxy)methyl]-7-amino-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid | C10H12N2O5S | 详情 | 详情 | |
| (II) | 69618 | (6R,7R)-7-amino-3-(hydroxymethyl)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid | C8H10N2O4S | 详情 | 详情 | |
| (III) | 21351 | 2-Hydroxybenzaldehyde;Salicylic aldehyde；2-Formylphenol;salicylaldehyde | 90-02-8 | C7H6O2 | 详情 | 详情 |
| (VIII) | 64882 | (6R,7R)-7-amino-8-oxo-3-vinyl-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid | 79349-82-9 | C9H10N2O3S | 详情 | 详情 |
| (IX) | 69619 | (Z)-S-benzo[d]thiazol-2-yl 2-(2-aminothiazol-4-yl)-2-((trityloxy)imino)ethanethioate | C31H22N4O2S3 | 详情 | 详情 |
Extended Information