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【结 构 式】 
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【药物名称】 【化学名称】Benzo[b]thiophene-2-boronic acid 【CA登记号】98437-23-1 【 分 子 式 】C8H7BO2S 【 分 子 量 】178.01879 |
【开发单位】Northwestern University (Originator) 【药理作用】Antibiotics, ANTIINFECTIVE THERAPY, beta-Lactam Enhancers, beta-Lactamase Inhibitors |
合成路线1
The reaction of benzo[b]thiophene (I) with triethyl borate by means of butyllithium gives benzo[b]thiophene-2-boronic acid diethyl ester (II), which is hydrolyzed to the target compound in acidic medium.
Extended Information